1. Chemogenomics
  2. AVPR1A

AVPR1A

NCBI gene ID HGNC ID UniProt ID SwissProt ID Description Protein family
552
895
P37288
V1AR_HUMAN
arginine vasopressin receptor 1A
GPCR

Compounds

Compound EUbOPEN ID Compound name Compound image SMILES / InChIKey Mode of action Main target Chem QC data available Incucyte cytotox data available Multiplex data available Other annotation data available
EUB0000389a
RELCOVAPTAN
Chemical structure of compound RELCOVAPTAN
COC1=C(OC)C=C(C=C1)S(=O)(=O)N1[C@@H](C(=O)N2CCC[C@H]2C(N)=O)[C@](O)(C2=C1C=CC(Cl)=C2)C1=CC=CC=C1Cl
CEBYCSRFKCEUSW-NAYZPBBASA-N
Antagonist
AVPR1A
Yes
Yes
No
Yes
EUB0000446a
TC OT 39
Chemical structure of compound TC OT 39
CN1N=CC2=C1NC1=CC=CC=C1N(C2)C(=O)C1=CC(C)=C(CNC(=O)N2CCC[C@H]2C(=S)N2CCCN(C)CC2)C=C1
KSNHHKZYKYNBEI-NDEPHWFRSA-N
Partial agonist
AVPR1A
,
AVPR2
,
OXTR
Yes
Yes
No
Yes