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Chemogenomics
BRD2@BD1

BRD2@BD1

NCBI gene ID HGNC ID UniProt ID SwissProt ID Description Protein family

BRD2_HUMAN

bromodomain containing 2

Bromodomain

Compounds

Compound EUbOPEN ID Compound name Compound image SMILES / InChIKey Mode of action Main target Chem QC data available Incucyte cytotox data available Multiplex data available Other annotation data available

EUB0000102c

I-BET151 (GSK1210151A)

Chemical structure of compound I-BET151 (GSK1210151A)

COc1cc2c(cc1-c1c(C)noc1C)ncc1nc(O)n([C@H](C)c3ccccn3)c12

VUVUVNZRUGEAHB-CYBMUJFWSA-N

,

,

,

,

,

,

,

No

No

EUB0000330a

(+)-JQ1

Chemical structure of compound (+)-JQ1

Cc1sc2c(c1C)C(c1ccc(Cl)cc1)=NC(CC(=O)OC(C)(C)C)c1nnc(C)n1-2

DNVXATUJJDPFDM-KRWDZBQOSA-N

,

,

,

,

,

,

,

No

No

The EUbOPEN project has received funding from the Innovative Medicines Initiative 2 Joint Undertaking under grant agreement No 875510. This Joint Undertaking receives support from the European Union's Horizon 2020 research and innovation programme, EFPIA companies and Associated Partners: KTH, OICR, Diamond and McGill. This communication reflects the views of the authors and neither IMI nor the European Union, EFPIA or any Associated Partners are liable for any use that may be made of the information contained herein.

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